Liste des publications, livres, chapitres de livre et brevets 2010-

Thématique Synthèse Organique

Publications

M. Belaud-Rotureau, T.T. Le, T.H.T. Phan, T.H. Nguyen, R. Aissaoui, F. Gohier, A. Derdour, A. Nourry, A.-S. Castanet, K.P.P. Nguyen, and J. Mortier, Synthesis of N-Aryl and N-Alkyl Anthranilic Acids via SNAr Reaction of Unprotected 2-Fluoro- and 2-Methoxybenzoic Acids by Lithioamides. Organic Letters, 2010. 12(10): p. 2406-2409.

S. Guillarme, J.-B. Behr, C. Bello, P. Vogel, and C. Saluzzo, Synthesis and glycosidase inhibitory activity of 1-amino-3,6-anhydro-1-deoxy-d-sorbitol derivatives. Bioorganic Chemistry, 2010. 38(2): p. 43-47.

K. Krohn, A. Vidal, H.T. Tran-Thien, U. Flörke, A. Bechthold, G. Dujardin, and I. Green, Total Synthesis of Silyl-Protected Early Intermediates of Polyketide Biosynthesis. European Journal of Organic Chemistry, 2010(16): p. 3080-3092.

T.T. Le, S. Guillarme, and C. Saluzzo, New class of [beta]-aminoalcohol ligands derived from isosorbide and isomannide: application in hydrogen transfer reduction of prochiral ketones. Tetrahedron, 2010. 66(46): p. 8893-8898.

C. Lucchesi, A. Arboré, S. Pascual, L. Fontaine, C. Maignan, and G. Dujardin, Solid-phase de novo synthesis of a (±)-2-deoxy-glycoside. Carbohydrate Research, 2010. 345(6): p. 844-849.

T.B. Nguyen, A. Beauseigneur, A. Martel, R. Dhal, M. Laurent, and G. Dujardin, Access to α-Substituted Amino Acid Derivatives via 1,3-Dipolar Cycloaddition of α-Amino Ester Derived Nitrones. The Journal of Organic Chemistry, 2010. 75(3): p. 611-620.

T.B. Nguyen, A. Martel, C. Gaulon, R. Dhal, and G. Dujardin, 1,3-Dipolar Cycloadditions of Nitrones to Heterosubstituted Alkenes. Part 1: Oxa and Aza-substituted Alkenes. Organic Preparations and Procedures International, 2010. 42(5): p. 387-432.

S. Pascual, T. Blin, P.J. Saikia, M. Thomas, P. Gosselin, and L. Fontaine, Block copolymers based on 2-vinyl-4,4-dimethyl-5-oxazolone by RAFT polymerization: Experimental and computational studies. Journal of Polymer Science Part A: Polymer Chemistry, 2010. 48(22): p. 5053-5062.

M.S.M. Pearson-Long, A. Beauseigneur, P. Karoyan, J. Szymoniak, and P. Bertus, Titanium-Catalyzed Cyclopropanation of Boc-Protected Cyanohydrins: A Short Access to Aminocyclopropanecarboxylic Acid Derivatives. Synthesis, 2010(20): p. 3410-3414.

P. Setzer, A. Beauseigneur, M.S.M. Pearson-Long, and P. Bertus, Titanium-Mediated Synthesis of 1,4-Diketones from Grignard Reagents and Acyl Cyanohydrins. Angewandte Chemie International Edition, 2010. 49(46): p. 8691-8694.

D. Tilly, J.-M. Fu, B.-P. Zhao, M. Alessi, A.-S. Castanet, V. Snieckus, and J. Mortier, On the Mechanism of the Directed ortho and Remote Metalation Reactions of N,N-Dialkylbiphenyl 2-carboxamides. Organic Letters, 2010. 12(1): p. 68-71.

A. Banchet-Cadeddu, A. Martinez, S. Guillarme, V. Parietti, F. Monneaux, E. Hénon, J.-H. Renault, J.-M. Nuzillard, and A. Haudrechy, Use of the NEO strategy (Nucleophilic addition/Epoxide Opening) for the synthesis of a new C-galactoside ester analogue of KRN 7000. Bioorganic & Medicinal Chemistry Letters, 2011. 21(8): p. 2510-2514.

S. Comesse, A. Martel, and A. Daïch, Domino Process Optimized via ab Initio Study for an Alternative Access to Bicyclic Lactams. Organic Letters, 2011. 13(15): p. 4004-4007.

S. Dalençon, R.A. Youcef, M. Pipelier, V. Maisonneuve, D. Dubreuil, F. Huet, and S. Legoupy, Asymmetric Synthesis of Cyclohexene Nucleoside Analogues. The journal of Organic Chemistry, 2011. 76(19): p. 8059-8063.

K. Guitot, M. Larregola, T.K. Pradhan, J.-L. Vasse, S. Lavielle, P. Bertus, J. Szymoniak, O. Lequin, and P. Karoyan, The Combination of Prolinoamino Acids and Cyclopropylamino Acids Leads to Fully Functionalized, Stable β-Turns in Water. ChemBioChem, 2011. 12(7): p. 1039-1042.

M.Y. Laurent, V. Stocker, V.M. Temgoua, G. Dujardin, and R. Dhal, New two-step sequence involving a hetero-Diels-Alder and a nonphenolic oxidative coupling reaction: a convergent access to analogs of steganacin. Tetrahedron Letters, 2011. 52(14): p. 1608-1611.

T.T. Le, N.T.T. Chau, T.T. Nguyen, J. Brien, T.T. Thai, A. Nourry, A.-S. Castanet, K.P.P. Nguyen, and J. Mortier, Evidence for a Trianion Intermediate in the Metalation of 4-Hydroxy-6,7-dimethoxy-8-methyl-2-naphthoic Acid. Methodology and Application to Racemic 5,5′-Didesisopropyl-5,5′-dialkylapogossypol Derivatives. The Journal of Organic Chemistry, 2011. 76(2): p. 601-608.

S. Leconte, A. Cena, A. Balquet, L. Cauret, T. Falher, D. Jouannet, R. Dhal, V. Montembault, P.-J. Madec, and C. Gondard, In-bulk formation of a new tetrasubstituted furan from phenolic antioxidants and dibasic lead stearate. Polymer Degradation and Stability, 2011. 96(4): p. 727-731.

N. Louaisil, P.D. Pham, F. Boeda, D. Faye, A.S. Castanet, and S. Legoupy, Ionic Liquid Supported Organotin Reagents: Green Tools for Stille CrossCoupling Reactions with Brominated Substrates. European Journal of Organic Chemistry, 2011. (1): p. 143-149.

J. Mortier, The Meyers Reaction (1994-2010). Current Organic Chemistry, 2011. 15(14): p. 2413-2437.

N.H. Nguyen, C. Len, A.-S. Castanet, and J. Mortier, Selectivity in C-alkylation of dianions of protected 6-methyluridine. Beilstein Journal of Organic Chemistry, 2011. 7: p. 1228-1233.

R. Aissaoui, A. Nourry, A. Coquel, T.T.H. Dao, A. Derdour, J.-J. Helesbeux, O. Duval, A.-S. Castanet, and J. Mortier, ortho-Lithium/Magnesium Carboxylate-Driven Aromatic Nucleophilic Substitution Reactions on Unprotected Naphthoic Acids. The journal of Organic Chemistry, 2012. 77(1): p. 718-724.

F. Boukattaya, A. Stanovych, P. Setzer, S. Abid, H. Ammar, M.S.M. Pearson-Long, and P. Bertus, Simple and convenient access to α,α,α-trisubstituted amides by double addition of Grignard reagents to acyl cyanohydrins. Chemical Communications, 2012. 48(69): p. 8655-8657.

D. Declerck, S. Josse, A. Nguyen Van Nhien, J. Szymoniak, P. Bertus, and D. Postel, Reactivity of sugar α-aminonitrile derivatives under titanium-mediated cyclopropanation conditions. Tetrahedron, 2012. 68(4): p. 1145-1152.

D. Declerck, A. Nguyen Van Nhien, S. Josse, J. Szymoniak, P. Bertus, C. Bello, P. Vogel, and D. Postel, Synthesis of 2-(1-aminocyclopropyl)pyrrolidine-3,4-diol derivatives applying titanium-mediated reaction conditions. Tetrahedron, 2012. 68(6): p. 1802-1809.

J. Hunault, M. Diswall, J.-C. Frison, V. Blot, J. Rocher, S. Marionneau-Lambot, T. Oullier, J.-Y. Douillard, S. Guillarme, C. Saluzzo, G. Dujardin, D. Jacquemin, J. Graton, J.-Y. Le Questel, M. Evain, J. Lebreton, D. Dubreuil, J. Le Pendu, and M. Pipelier, 3-Fluoro- and 3,3-Difluoro-3,4-dideoxy-KRN7000 Analogues as New Potent Immunostimulator Agents: Total Synthesis and Biological Evaluation in Human Invariant Natural Killer T Cells and Mice. The journal of Medicinal Chemistry, 2012. 55(3): p. 1227-1241.

A. Lancou, H. Haroun, U.K. Kundu, F. Legros, N. Zimmermann, M. Mathé-Allainmat, J. Lebreton, G. Dujardin, C. Gaulon-Nourry, and P. Gosselin, α-Triethylsilyl-α-diazoacetone in double cross-aldolisation: convenient acetone equivalent toward 5-hydroxy-1,3-diketones. Tetrahedron, 2012. 68(47): p. 9652-9657.

D. Le, V. Montembault, S. Pascual, S. Legoupy, and L. Fontaine, An Orthogonal Modular Approach to Macromonomers Using Clickable Cyclobutenyl Derivatives and RAFT Polymerization. Macromolecules, 2012. 45(19): p. 7758-7769.

T.B. Nguyen, A. Martel, C. Gaulon-Nourry, R. Dhal, and G. Dujardin, 1,3-Dipolar Cycloadditions of Nitrones to Hetero-substituted Alkenes Part 2: Sila-, Thia-, Phospha- and Halo-substituted Alkenes. Organic Preparations and Procedures International, 2012. 44(1): p. 1-81.

K.B. Selim, A. Beauchard, J. Lhoste, A. Martel, M.Y. Laurent, and G. Dujardin, Organocatalytic enantio- and diastereoselective 1,3-dipolar cycloaddition between alanine-derived ketonitrones and E-crotonaldehyde: efficiency and full stereochemical studies. Tetrahedron: Asymmetry, 2012. 23(24): p. 1670-1677.

P. Shpak-Kraievskyi, B. Yin, A. Martel, R. Dhal, G. Dujardin, and M.Y. Laurent, Access to C-protected β-amino-aldehydes via transacetalization of 6-alcoxy tetrahydrooxazinones and use for pseudo-peptide synthesis. Tetrahedron, 2012. 68(9): p. 2179-2188.

D. Tilly, J. Magolan, and J. Mortier, Directed Remote Aromatic Metalations: Mechanisms and Driving Forces. Chemistry – A European Journal, 2012. 18(13): p. 3804-3820.

J. Totobenazara, H. Haroun, J. Rémond, K. Adil, F. Dénès, J. Lebreton, C. Gaulon-Nourry, and P. Gosselin, Tandem Payne/Meinwald versus Meinwald rearrangements on the α-hydroxy- or α-silyloxy-spiro epoxide skeleton. Organic & Biomolecular Chemistry, 2012. 10(3): p. 502-505.

C.S. Vu, N. Guisot, S. Guillarme, A. Martel, G. Dujardin, M. Pipelier, D. Dubreuil, and C. Saluzzo, A Convergent Hetero-Diels–Alder Strategy for Asymmetric Access to a Lactone Containing Two Lipidic Chains. European Journal of Organic Chemistry, 2012. (20): p. 3727-3731.

A. Boussonnière, R. Bénéteau, J. Lebreton, and F. Dénès, Aluminum Acetals in Organic Synthesis. European Journal of Organic Chemistry, 2013. (35): p. 7853-7866.

L.-Y. Chen, S. Guillarme, and C. Saluzzo, Dianhydrohexitols: new tools for organocatalysis. Application in enantioselective Friedel-Crafts alkylation of indoles with nitroalkenes. ARKIVOC, 2013. 3: p. 227-244.

D. Faye, M. Vybornyi, F. Boeda, and S. Legoupy, Solvent free hydrostannation and Stille reactions using ionic liquid supported organotin reagents. Tetrahedron, 2013. 69(26): p. 5421-5425.

D. Le, G. Morandi, S. Legoupy, S. Pascual, V. Montembault, and L. Fontaine, Cyclobutenyl macromonomers: Synthetic strategies and ring-opening metathesis polymerization. European Polymer Journal, 2013. 49(5): p. 972-983.

B. Oberleitner, A. Dellinger, M. Deforet, A. Galtayries, A.-S. Castanet, and V. Semetey, A facile and versatile approach to design self-assembled monolayers on glass using thiol-ene chemistry. Chemical Communications, 2013. 49(16): p. 1615-1617.

C. Szalata, J. Szymoniak, F. Fabis, S. Butt-Gueulle, S. Rault, P. Bertus, S. Gérard, and J. Sapi, Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT(6) Receptor Ligands. ChemMedChem, 2013. 8(1): p. 70-73.

N. Zimmermann, P. Pinard, B. Carboni, P. Gosselin, C. Gaulon-Nourry, G. Dujardin, S. Collet, J. Lebreton, and M. Mathé-Allainmat, Convergent Strategy Towards the Synthesis of Restricted Analogues of Peloruside A. European Journal of Organic Chemistry, 2013. (12): p. 2303-2315.

K. Ben Ayed, A. Beauchard, J.-F. Poisson, S. Py, M.Y. Laurent, A. Martel, H. Ammar, S. Abid, and G. Dujardin, Asymmetric Access to α-Substituted Functional Aspartic Acid Derivatives by a [3+2] Strategy Employing a Chiral Dienophile. European Journal of Organic Chemistry, 2014. (14): p. 2924-2932.

L.Y. Chen, S. Guillarme, A. Whiting, and C. Saluzzo, Asymmetric Michael addition of acetone to beta-nitrostyrenes catalyzed by novel organocatalysts derived from D-isomannide or L-isoidide. ARKIVOC, 2014: p. 215-227.

G. Darmograi, L. Jouffret, A. Hémon-Ribaud, M. Leblanc, G. Dujardin, V. Maisonneuve, and J. Lhoste, Fluoroferrates with (dabcoH2)2+ or (dabcoH)+ Cations. Journal of Inorganic and General Chemistry, 2014. 640(7): p. 1385-1391.

E. Maougal, S. Dalençon, M.S.M. Pearson-Long, M. Mathé-Allainmat, J. Lebreton, and S. Legoupy, An Efficient Synthesis of 3,3′-Bipiperidines Using an ROM/RCM Metathesis Sequence: Extension to Oxygenated Analogues. Synthesis, 2014. 46(23): p. 3268-3272.

T.T.T. Nguyen, A. Boussonnière, E. Banaszak, A.-S. Castanet, K.P.P. Nguyen, and J. Mortier, Chemoselective Deprotonative Lithiation of Azobenzenes: Reactions and Mechanisms. The Journal of Organic Chemistry, 2014. 79(6): p. 2775-2780.

K.B. Selim, A. Martel, M.Y. Laurent, J. Lhoste, S. Py, and G. Dujardin, Enantioselective Ruthenium-Catalyzed 1,3-Dipolar Cycloadditions between C-Carboalkoxy Ketonitrones and Methacrolein: Solvent Effect on Reaction Selectivity and Its Rational. The Journal of Organic Chemistry, 2014. 79(8): p. 3414-3426.

P. Setzer, G. Forcher, F. Boeda, M.S.M. Pearson-Long, and P. Bertus, Titanium-Mediated Addition of Grignard Reagents to Acyl Cyanohydrins: Aminocyclopropane versus 1,4-Diketone Formation. European Journal of Organic Chemistry, 2014. (1): p. 171-180.

X. Zhang, P. Cividino, J.-F. Poisson, P. Shpak-Kraievskyi, M.Y. Laurent, A. Martel, G. Dujardin, and S. Py, Asymmetric Synthesis of α,α-Disubstituted Amino Acids by Cycloaddition of (E)-Ketonitrones with Vinyl Ethers. Organic Letters, 2014. 16(7): p. 1936-1939.

I. Abid, P. Gosselin, M. Mathé-Allainmat, S. Abid, G. Dujardin and C. Gaulon-Nourry, TBAF-triggered aldol-type addition of a-triethylsilyl-a-diazoacetone. The Journal of Organic Chemistry, 2015 80(20): p. 9980–9988.

M. Berthet, F. Davanier, G. Dujardin, J. Martinez and I. Parrot, MgI2-mediated Chemoselective Cleavage of Protecting Groups, an Alternative to Conventional Deprotection Methodologies. Chemistry – A European Journal, 2015, 21(31): p. 11014-11016.

G. Forcher, N. Clousier, A. Beauseigneur, P. Setzer, F. Boeda, M.S.M. Pearson-Long, P. Karoyan, J. Szymoniak, and P. Bertus, Titanium-Mediated Cyclopropanation of Nitriles with Unsaturated Grignard Reagents: Application to the Synthesis of Constrained Lysine Derivatives. Synthesis, 2015. 47(7): p. 992-1006.

G. Forcher, A. Silvanus, P. de Frémont, B. Jacques, M.S.M. Pearson-Long, F. Boeda, and P. Bertus, A stereoselective access to a ferrocene-based planar chiral triazolium salt. The Journal of Organometallic Chemistry, 2015 797 : p. 1-7.

M. Kadraoui, T. Maunoury, Z. Derriche, S. Guillarme, and C. Saluzzo, Isohexides as Versatile Scaffolds for Asymmetric Catalysis. European Journal of Organic Chemistry, 2015. (3): p. 441-457.

R. Le Goff, A. Martel, M. Sanselme, A.M. Lawson, A. Daïch, and S. Comesse, Simple Access to Highly Functional Bicyclic γ- and δ-Lactams: Origins of Chirality Transfer to Contiguous Tertiary/Quaternary Stereocenters Assessed by DFT. Chemistry – A European Journal, 2015. 21(7): p. 2966-2979.

N. Le Marquer, M.Y. Laurent, and A. Martel, A practical and cost effective method for bicyclo[2.2.2]octane-1,4-dicarboxylic acid synthesis. Synthesis, 2015. 47(15): p. 2185-2187.

T.T.T. Nguyen, G. Contrel, V. Montembault, G. Dujardin, and L. Fontaine, Phosphonated furan-functionalized poly(ethylene oxide)s using orthogonal click chemistries: synthesis and Diels-Alder reactivity. Polymer Chemistry, 2015. 6(16): p. 3024-3030.

V. Pimenta, Q.H.H. Le, L. Clark, J. Lhoste, A. Hemon-Ribaud, M. Leblanc, J.-M. Greneche, G. Dujardin, P. Lightfoot, and V. Maisonneuve, New iron tetrazolate frameworks: synthesis, temperature effect, thermal behaviour, Mossbauer and magnetic studies. Dalton Transactions, 2015. 44(17): p. 7951-7959.

V. Pimenta, J. Lhoste, A. Hemon-Ribaud, M. Leblanc, J.-M. Greneche, L. Jouffret, A. Martel, G. Dujardin and V. Maisonneuve, Evidence of new fluorinated coordination compounds in the composition space diagram of FeF3/ZnF2-Hamtetraz-HFaq. System. Crystal Growth & Design, 2015 15(9): pp 4248–4255

P. Shpak-Kraievskyi, A. Mankou Makaya, A. Beauchard, A. Martel, M.Y. Laurent, and G. Dujardin, [3+2] Route to Quaternary Oxaprolinol Derivatives as Masked Precursors of Disubstituted β33-Amino Aldehyde. European Journal of Organic Chemistry, 2015 81(6): p. 3923-3934.

M. Belaud-Rotureau, A.-S. Castanet, T. H. Nguyen and J.  Mortier, Uncatalyzed CO2Li-Mediated SNAr Reaction of Unprotected Benzoic Acids via Silicon Trickery. Australian Journal of Chemistry, 2016 69(3): p. 307-313. 

F. Boukattaya, J. Caillé, H. Ammar, F. Rouzier, F. Boeda, M. Pearson-Long, P Bertus, A short Access to Symmetrically α,α-Disubstituted α-Amino Acids from Acyl Cyanohydrin Synthesis 2016, 48 : p. 906-916.

T. Chalopin, K. Jebali, C. Gaulon-Nourry, F. Dénès, J., M. Mathé-Allainmat Regioselective dihydropyran formation from 4-iodo-2,6-disubstituted tetrahydropyran derivatives using In(OAc)3/LiI system as the promoter Tetrahedron 2016, 72 : p. 318-327.

A. El Bouakher, R. Le Goff, J. Tasserie, J. Lhoste, A. Martel, S. Comesse Synthesis of Oxazolidin-4-ones: Domino O-Alkylation/Aza-Michael/Intramolecular Retro-Claisen Condensation Organic Letters 2016 18(10): p. 2383-2386.

M. Berthet; T. Cheviet; G. Dujardin; I. Parrot; J. Martinez Isoxazolidine: A Privileged Scaffold for Organic and Medicinal Chemistry. Chem. Rev. 2016, 116 (24), 15235-15283.

N. E. S. Guisot; I. Ella Obame; P. Ireddy; A. Nourry; C. Saluzzo; G. Dujardin; D. Dubreuil; M. Pipelier; S. Guillarme Reaction of Glyconitriles with Organometallic Reagents: Access to Acyl β-C-Glycosides. J. Org. Chem.2016, 81 (6), 2364-2371.

A. Hamdi; A. S. Mostafa; C. N. Watat; M. Y. Laurent; K. Ben Ayed; K. B. Selim; G. Dujardin Acetylene-free synthesis of vinyloxy pyridine and quinoline. Tetrahedron Lett.2016, 57 (51), 5825-5829.

I. Abid; S. Gavelle; A.-C. Chany; F. Legros; P. Gosselin; S. Abid; G. Dujardin; C. Gaulon-Nourry Advances in the TBAF-induced aldol-type addition of α-trialkylsilyl-α-diazoacetones: TIPS versus TES. C. R. Chim.2017, Ahead of Print.

M. S. M. Pearson-Long; F. Boeda; P. Bertus Double Addition of Organometallics to Nitriles: Toward an Access to Tertiary Carbinamines. Adv. Synth. Catal.2017, 359 (2), 179-201.

 

Livres/Chapitres de livres

C. Saluzzo and S. Guillarme, Nitrogen-Containing Ligands Anchored onto Polymers as Catalyst Stabilizer for Catalytic Enantioselective Reactions, Advances in Chemistry Ressearch, 2010. 3: p.257-388.

C. Saluzzo and S. Guillarme, Nitrogen-Containing Ligands Anchored onto Polymers as Catalyst Stabilizer for Catalytic Enantioselective Reactions, in Polymer Aging, Stabilizers and Amphiphilic Polymer Block Copolymers, L. Segewicz and M. Petrowsky, Editors. Chapter 3. 2011, Editions Nova Science Publishers

C. Saluzzo and S. Guillarme, Nitrogen-Containing Ligands Anchored onto Polymers as Catalyst Stabilizer for Catalytic Enantioselective Reactions, in Encyclopedia of Polymer Research, C.E. Jones, Editor. 2011, Editions Nova Science Publishers, p.45-172.

C. Saluzzo and S. Guillarme, Asymmetric heterogeneous supported catalysis: use of nitrogen-containing ligands. 2012, Editions Nova Science Publishers.

P. Bertus, F. Boeda, and M.S.M. Pearson-Long, Titanium-Mediated Synthesis of Cyclopropyl Derivatives, in Science of Synthesis Knowledge Updates, J.J. Li, I. Marek, M. North, M. Oestreich, E. Schaumann, S.M. Weinreb and M. Yus, Editors. Vol. 1. 2012, Editions Stuttgart : London, Georg Thieme Verlag. p. 1-50.

A.-S. Castanet, A. Boussonnière, and J. Mortier, Asymmetric Nucleophilic Aromatic Substitution, in Arene Chemistry: Reaction Mechanisms and Methods for Aromatic Compounds, J. Mortier, Editor. 2015, Editions John Wiley and sons, Inc. Haubauken N.J.

J. Mortier and F. Leroux, Directed Metalation of Arenes with Organolithiums, Lithium Amides, and Superbases, in Arene Chemistry: Reaction Mechanisms and Methods for Aromatic Compounds, J. Mortier, Editor. 2015, Editions John Wiley and sons, Inc. Haubauken N.J.

P. Bertus, F. Boeda, and M.S.M. Pearson-Long, Titanium Based Catalysts for Asymmetric Transformations, in Sustainable Catalysis: With Non-endangered Metals, Part 1, The Royal Society of Chemistry: 2016; pp 140-198.

 

Brevets

Gossypol and apogossypol derivatives, preparation thereof and use thereof, J. Mortier, A.-S. Castanet, N.T.T. Chau. US Patent US8455540B2 (2013), US20100331398A1 (2010), EP Patent EP2231573 (2010).

Method for Preparing Chemical Compounds of Interest by Nucleophilic Aromatic Substitution of Aromatic Carboxylic Acid Derivatives Supporting at Least One Electro-Attractive Group, J. Mortier, A.-S. Castanet, A. Nourry, M. Belaud-Rotureau, WO Patent WO2011101604A1 (2011), US Patent US2012316337A1 (2012), FR Patent FR2961204 (2011).

Method for Preparing Chemical Compounds of Interest by Aromatic Nucleophilic Substitution, J. Mortier, A.-S. Castanet, M. Belaud-Rotureau, WO Patent WO2011101599A1 (2011),  US2012316337A1 (2012), FR Patent FR2956662A1 (2011).

Procédé de préparation d’omega-alcynylsilane, J. Mortier, A.-S. Castanet, E. Banaszak, FR Patent FR2942228A1 (2010).

Ionic liquid supported organotin reagents for the manufacturing of radiopharmaceuticals compounds, F. Boeda, A. Faivre-Chauvet, D. Faye, J.-F. Gestin, S. Legoupy, H. Rajerison, EP Patent EP 14150296.3-1451 (2014). Extension PCT/EP2015/050180 (2015).

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